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PNU-177864 hydrochloride

CAS No. 1783978-03-9

PNU-177864 hydrochloride ( PNU-177864 (hydrochloride) )

产品货号. M26387 CAS No. 1783978-03-9

PNU-177864 hydrochloride is a selective antagonist of D3 receptor with antischizophrenic activity.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥405 有现货
10MG ¥608 有现货
25MG ¥1037 有现货
50MG ¥1555 有现货
100MG ¥2325 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    PNU-177864 hydrochloride
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    PNU-177864 hydrochloride is a selective antagonist of D3 receptor with antischizophrenic activity.
  • 产品描述
    PNU-177864 hydrochloride is a selective antagonist of D3 receptor with antischizophrenic activity.(In Vivo):In Sprague-Dawley rats, PNU-177864 hydrochloride (8-200 mg/kg; gavage) induces phospholipidosis in unusual target organs including epididymis, hair follicles and pituitary.
  • 同义词
    PNU-177864 (hydrochloride)
  • 通路
    GPCR/G Protein
  • 靶点
    Dopamine Receptor
  • 受体
    VHL
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1783978-03-9
  • 分子量
    438.9
  • 分子式
    C18H22ClF3N2O3S
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    Cl.O=S(=O)(NC1=CC=C(C=C1)CCNCCC)C2=CC=C(OC(F)(F)F)C=C2
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562.
产品手册
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