
PNU-177864 hydrochloride
CAS No. 1783978-03-9
PNU-177864 hydrochloride ( PNU-177864 (hydrochloride) )
产品货号. M26387 CAS No. 1783978-03-9
PNU-177864 盐酸盐是一种选择性 D3 受体拮抗剂,具有抗精神分裂症活性。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥405 | 有现货 |
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10MG | ¥608 | 有现货 |
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25MG | ¥1037 | 有现货 |
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50MG | ¥1555 | 有现货 |
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100MG | ¥2325 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称PNU-177864 hydrochloride
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述PNU-177864 盐酸盐是一种选择性 D3 受体拮抗剂,具有抗精神分裂症活性。
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产品描述PNU-177864 hydrochloride is a selective antagonist of D3 receptor with antischizophrenic activity.(In Vivo):In Sprague-Dawley rats, PNU-177864 hydrochloride (8-200 mg/kg; gavage) induces phospholipidosis in unusual target organs including epididymis, hair follicles and pituitary.
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体外实验——
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体内实验PNU-177864 (12.5-200 mg/kg; oral gavage; daily; for 2-4 weeks; Sprague-Dawley rats) treatment induces phospholipidosis in unusual target organs in dogs or rats including epididymis, pituitary, and hair follicles. Animal Model:Male and female Sprague-Dawley rats (8-9-week-old)Dosage:12.5 mg/kg, 50 mg/kg (for 2 weeks), or 200 mg/kg; 8 mg/kg, 25 mg/kg, or 80 mg/kg (for 4 weeks)Administration:Oral gavage; daily; for 2-4 weeks Result:Induced phospholipidosis in unusual target organs in dogs or rats including epididymis, pituitary, and hair follicles.
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同义词PNU-177864 (hydrochloride)
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通路GPCR/G Protein
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靶点Dopamine Receptor
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受体VHL
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研究领域——
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适应症——
化学信息
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CAS Number1783978-03-9
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分子量438.89
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分子式C18H22ClF3N2O3S
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纯度>98% (HPLC)
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溶解度——
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SMILESCl.O=S(=O)(NC1=CC=C(C=C1)CCNCCC)C2=CC=C(OC(F)(F)F)C=C2
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562.
产品手册




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